Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Endoplasmin (Homo sapiens (Human)) | BDBM126083 (US8779142, 102) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to GRP94 (unknown origin) by fluorescence polarization competitive binding assay | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01715 BindingDB Entry DOI: 10.7270/Q2Z323H2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endoplasmin (Homo sapiens (Human)) | BDBM126083 (US8779142, 102) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
China Pharmaceutical University Curated by ChEMBL | Assay Description Inhibition of FITC-geldanamycin binding to N-terminal His-tagged recombinant human GRP94 expressed in Escherichia coli preincubated for 2 hrs followe... | J Med Chem 63: 1798-1822 (2020) Article DOI: 10.1021/acs.jmedchem.9b00940 BindingDB Entry DOI: 10.7270/Q23X8B3C | |||||||||||
More data for this Ligand-Target Pair |