Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Endothelin-1 receptor (Homo sapiens (Human)) | BDBM50071448 (CHEMBL307033 | N-[(S)-1-[(S)-1-(Butane-1-sulfonyla...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 6.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takarazuka Research Institute Curated by ChEMBL | Assay Description Compound was tested for the binding affinity against Endothelin A receptor | Bioorg Med Chem Lett 8: 2247-52 (1999) BindingDB Entry DOI: 10.7270/Q26M3609 | |||||||||||
More data for this Ligand-Target Pair |