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Found 1 hit Enz. Inhib. hit(s) with Target = 'Fatty-acid amide hydrolase 1' and Ligand = 'BDBM50174997'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Fatty-acid amide hydrolase 1


(Homo sapiens (Human))		BDBM50174997
PNG
(CHEMBL3809683)
Show SMILES Clc1ccc(Oc2cccc(CC3CCN(CC3)C(=O)Nc3cccnc3)c2)nc1
Show InChI InChI=1S/C23H23ClN4O2/c24-19-6-7-22(26-15-19)30-21-5-1-3-18(14-21)13-17-8-11-28(12-9-17)23(29)27-20-4-2-10-25-16-20/h1-7,10,14-17H,8-9,11-13H2,(H,27,29)
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Similars
Article
PubMed
n/an/a 1n/an/an/an/an/an/a



Janssen Pharmaceutical Companies of Johnson& Johnson, L.L.C.

Curated by ChEMBL


Assay Description
Apparent inhibition of recombinant human FAAH expressed in SK-N-MC cells assessed as [3H]-anandamide hydrolysis after 1 hr by liquid scintillation an...

Bioorg Med Chem Lett 26: 3109-14 (2016)


Article DOI: 10.1016/j.bmcl.2016.05.001
BindingDB Entry DOI: 10.7270/Q25B04F3
More data for this
Ligand-Target Pair