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Found 1 hit Enz. Inhib. hit(s) with Target = 'Fatty-acid amide hydrolase 1 [30-579]' and Ligand = 'BDBM50242674'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Fatty-acid amide hydrolase 1 [30-579]


(Rattus norvegicus (rat))
BDBM50242674
PNG
(5-((4-azido-3-iodobenzamido)methyl)-N,N-dimethyl-2...)
Show SMILES CN(C)C(=O)n1nnc(CNC(=O)c2ccc(N=[N+]=[N-])c(I)c2)n1
Show InChI InChI=1S/C12H12IN9O2/c1-21(2)12(24)22-18-10(17-20-22)6-15-11(23)7-3-4-9(16-19-14)8(13)5-7/h3-5H,6H2,1-2H3,(H,15,23)
PDB
MMDB

UniProtKB/SwissProt

B.MOAD
GoogleScholar
AffyNet 
CHEMBL
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 25n/an/an/an/an/an/a



Università di Roma La Sapienza

Curated by ChEMBL


Assay Description
Inhibition of FAAH mediated [14C]anadamide hydrolysis in rat brain after 30 mins


Eur J Med Chem 43: 62-72 (2008)


Article DOI: 10.1016/j.ejmech.2007.02.023
BindingDB Entry DOI: 10.7270/Q2154GS8
More data for this
Ligand-Target Pair