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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Fibroblast growth factor receptor 2 [400-821]' and Ligand = 'BDBM436198'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Fibroblast growth factor receptor 2 [400-821]


(Homo sapiens (Human))		BDBM436198
PNG
(US10590109, Compound 16)
Show SMILES CC(C)Nc1cc(NC(=O)N(C)c2ccc(CN3CCN(C)CC3=O)c(C=O)n2)ncc1C#N
Show InChI InChI=1S/C23H28N8O3/c1-15(2)26-18-9-20(25-11-17(18)10-24)28-23(34)30(4)21-6-5-16(19(14-32)27-21)12-31-8-7-29(3)13-22(31)33/h5-6,9,11,14-15H,7-8,12-13H2,1-4H3,(H2,25,26,28,34)
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a>1.00E+3n/an/an/an/an/an/a



Nanjing InnoCare Pharma Tech Co., Ltd.

US Patent


Assay Description
FGFR2: The in vitro activity of FGFR2 was determined by assaying the phosphorylation level of the substrate in the kinase reaction, by means of an HT...

US Patent US10590109 (2020)


BindingDB Entry DOI: 10.7270/Q2J969D2
More data for this
Ligand-Target Pair