Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Free fatty acid receptor 4 (Homo sapiens (Human)) | BDBM50203660 (CHEMBL3896714) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 290 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR120 expressed in CHOK1 cells measured after 60 mins by IP1-HTRF assay | Bioorg Med Chem Lett 26: 5724-5728 (2016) Article DOI: 10.1016/j.bmcl.2016.10.054 BindingDB Entry DOI: 10.7270/Q24Q7WZ2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 4 (Mus musculus) | BDBM50203660 (CHEMBL3896714) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 140 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR120 expressed in CHOK1 cells measured after 60 mins by IP1-HTRF assay | Bioorg Med Chem Lett 26: 5724-5728 (2016) Article DOI: 10.1016/j.bmcl.2016.10.054 BindingDB Entry DOI: 10.7270/Q24Q7WZ2 | |||||||||||
More data for this Ligand-Target Pair |