BindingDB PrimarySearch

Found 2 hits Enz. Inhib. hit(s) with Target = 'Free fatty acid receptor 4' and Ligand = 'BDBM50386790'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Free fatty acid receptor 4 (Homo sapiens (Human))	BDBM50386790 (CHEMBL1829174 \| CHEMBL2047159 \| TAK-875 \| US119052...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid PDB UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a
Guangdong Pharmaceutical University Curated by ChEMBL					Assay Description Agonist activity at human FFAR4 expressed in CHO cells assessed as beta-arrestin recruitment after 90 mins by luminescence assay				Bioorg Med Chem 25: 6647-6652 (2017) Article DOI: 10.1016/j.bmc.2017.10.040 BindingDB Entry DOI: 10.7270/Q2Z3226M
Guangdong Pharmaceutical University Curated by ChEMBL					More data for this Ligand-Target Pair
Free fatty acid receptor 4 (Homo sapiens (Human))	BDBM50386790 (CHEMBL1829174 \| CHEMBL2047159 \| TAK-875 \| US119052...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid PDB UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Agonist activity at human GPR120 expressed in CHO cells assessed as calcium influx after 30 mins by FLIPR assay				ACS Med Chem Lett 1: 290-294 (2010) Article DOI: 10.1021/ml1000855 BindingDB Entry DOI: 10.7270/Q29G5NZJ
TBA Curated by ChEMBL					More data for this Ligand-Target Pair