Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
G-protein coupled receptor 183 (Homo sapiens (Human)) | BDBM50558426 (CHEMBL4788348) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | n/a | 0.0320 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at Go2-q-coupled human EBI2 expressed in COS7 cell membranes assessed as stimulation of [35S]GTPgammaS binding preincubated for 20 m... | Citation and Details Article DOI: 10.1016/j.bmcl.2016.09.029 BindingDB Entry DOI: 10.7270/Q2SX6HW6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
G-protein coupled receptor 183 (Homo sapiens (Human)) | BDBM50558426 (CHEMBL4788348) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | n/a | 0.140 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at Go2-q-coupled EBI2 (unknown origin) expressed in COS7 cell membranes assessed as stimulation of [35S]GTPgammaS binding preincubat... | Citation and Details Article DOI: 10.1016/j.bmcl.2016.09.029 BindingDB Entry DOI: 10.7270/Q2SX6HW6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
G-protein coupled receptor 183 (Mus musculus) | BDBM50558426 (CHEMBL4788348) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | n/a | 0.702 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at Go2-q-coupled mouse EBI2 expressed in COS7 cell membranes assessed as stimulation of [35S]GTPgammaS binding preincubated for 20 m... | Citation and Details Article DOI: 10.1016/j.bmcl.2016.09.029 BindingDB Entry DOI: 10.7270/Q2SX6HW6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
G-protein coupled receptor 183 (Rattus norvegicus) | BDBM50558426 (CHEMBL4788348) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | n/a | 1.30 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at Go2-q-coupled rat EBI2 expressed in COS7 cell membranes assessed as stimulation of [35S]GTPgammaS binding preincubated for 20 min... | Citation and Details Article DOI: 10.1016/j.bmcl.2016.09.029 BindingDB Entry DOI: 10.7270/Q2SX6HW6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) |