Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Gamma-aminobutyric acid receptor subunit alpha-1 (Homo sapiens (Human)) | BDBM98558 (US8492408, 7a) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Aniona APS US Patent | Assay Description In vitro inhibition assay using GABA receptor. | US Patent US8492408 (2013) BindingDB Entry DOI: 10.7270/Q28K77QX | |||||||||||
More data for this Ligand-Target Pair |