Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Gastrin/cholecystokinin type B receptor (Homo sapiens (Human)) | BDBM50092405 ((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-((S)-2-{[...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | 0.280 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Binding affinity against cholecystokinin type B receptor on guinea pig cortex. | J Med Chem 43: 3614-23 (2000) BindingDB Entry DOI: 10.7270/Q2RN373C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (RAT) | BDBM50092405 ((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-((S)-2-{[...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | 0.75 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Compound was tested for binding affinity against Cholecystokinin type B receptor expressed in CHO cells on the rat brain. | J Med Chem 43: 3614-23 (2000) BindingDB Entry DOI: 10.7270/Q2RN373C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (RAT) | BDBM50092405 ((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-((S)-2-{[...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | >3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Ability to displace 1 nM [3H]pCCK-8 from rat Cholecystokinin type B receptor stably expressing in CHO cells | Bioorg Med Chem Lett 14: 369-72 (2003) BindingDB Entry DOI: 10.7270/Q2RJ4K1Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastrin/cholecystokinin type B receptor (RAT) | BDBM50092405 ((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-((S)-2-{[...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | n/a | 0.400 | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain. | J Med Chem 43: 3614-23 (2000) BindingDB Entry DOI: 10.7270/Q2RN373C | |||||||||||
More data for this Ligand-Target Pair |