BindingDB logo
myBDB logout
Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Glucagon receptor' and Ligand = 'BDBM50244075'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Glucagon receptor


(Homo sapiens (Human))		BDBM50244075
PNG
(1-(3-chloro-4-(4-chlorophenoxy)phenyl)-3-(2-chloro...)
Show SMILES Clc1ccc(Oc2ccc(NC(=O)NC(=O)c3ccccc3Cl)cc2Cl)cc1
Show InChI InChI=1S/C20H13Cl3N2O3/c21-12-5-8-14(9-6-12)28-18-10-7-13(11-17(18)23)24-20(27)25-19(26)15-3-1-2-4-16(15)22/h1-11H,(H2,24,25,26,27)
PDB
MMDB

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
CHEMBL
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 482n/an/an/an/an/an/a



Merck Research Laboratories

Curated by ChEMBL


Assay Description
Displacement of [125I]glucagon from human GCGR expressed in CHO cells

Bioorg Med Chem Lett 18: 3701-5 (2008)


Article DOI: 10.1016/j.bmcl.2008.05.072
BindingDB Entry DOI: 10.7270/Q26Q1X25
More data for this
Ligand-Target Pair