Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Glucagon-like peptide 1 receptor (Homo sapiens (Human)) | BDBM349710 (2-[(4-{6-[(4-cyano-2-fluorobenzyl)oxy]pyridin-2-yl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 8.80 | n/a | n/a | n/a | n/a |
Pfizer Inc. US Patent | Assay Description GLP-1R-mediated agonist activity was determined with a cell-based functional assay utilizing an HTRF (Homogeneous Time-Resolved Fluorescence) cAMP de... | US Patent US10208019 (2019) BindingDB Entry DOI: 10.7270/Q2WH2S4X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon-like peptide 1 receptor (Homo sapiens (Human)) | BDBM349710 (2-[(4-{6-[(4-cyano-2-fluorobenzyl)oxy]pyridin-2-yl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 0.760 | n/a | n/a | n/a | n/a |
Pfizer Inc. US Patent | Assay Description GLP-1R-mediated agonist activity was determined with a cell-based functional assay utilizing an HTRF (Homogeneous Time-Resolved Fluorescence) cAMP de... | US Patent US10208019 (2019) BindingDB Entry DOI: 10.7270/Q2WH2S4X | |||||||||||
More data for this Ligand-Target Pair |