Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Glucose-dependent insulinotropic receptor' and Ligand = 'BDBM50036669'   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Glucose-dependent insulinotropic receptor (Homo sapiens (Human))	BDBM50036669 (CHEMBL3354800) Show SMILES COC(=O)[C@@]1(Cc2cccc(F)c2)NCc2cnc3c(c(nn3c12)C(C)(C)O)-c1ccc(cc1)C(F)(F)F |r| Show InChI InChI=1S/C27H24F4N4O3/c1-25(2,37)21-20(16-7-9-18(10-8-16)27(29,30)31)23-32-13-17-14-33-26(24(36)38-3,22(17)35(23)34-21)12-15-5-4-6-19(28)11-15/h4-11,13,33,37H,12,14H2,1-3H3/t26-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	n/a	n/a	530	n/a	n/a	n/a	n/a
Genomics Institute of the Novartis Research Foundation Curated by ChEMBL					Assay Description Agonist activity at human GPR119 overexpressed in CHO cells assessed as increase in cellular cAMP production by HTRF method				Bioorg Med Chem Lett 24: 5478-83 (2015) Article DOI: 10.1016/j.bmcl.2014.10.010 BindingDB Entry DOI: 10.7270/Q29C7019
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