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Found 1 hit Enz. Inhib. hit(s) with Target = 'Glucose-dependent insulinotropic receptor' and Ligand = 'BDBM50244684'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Glucose-dependent insulinotropic receptor


(Homo sapiens (Human))		BDBM50244684
PNG
(CHEMBL459873 | N-(4-(ethylsulfonyl)phenyl)-6-(4-(3...)
Show SMILES CCS(=O)(=O)c1ccc(Nc2ncnc(N3CCC(CC3)c3nc([n-][o+]3)C(C)C)c2[N+]([O-])=O)cc1
Show InChI InChI=1S/C22H27N7O5S/c1-4-35(32,33)17-7-5-16(6-8-17)25-20-18(29(30)31)21(24-13-23-20)28-11-9-15(10-12-28)22-26-19(14(2)3)27-34-22/h5-8,13-15H,4,9-12H2,1-3H3,(H,23,24,25)
PDB

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PC cid
PC sid
UniChem

Similars
Article
PubMed
n/an/an/an/a 17n/an/an/an/a



Arena Pharmaceuticals

Curated by ChEMBL


Assay Description
Agonist activity at CPR119 (unknown origin) transfected in Xenopus dermal melanophore assessed as dispersion of melatonin-induced pigmentation

J Med Chem 51: 5172-5 (2008)


Article DOI: 10.1021/jm8006867
BindingDB Entry DOI: 10.7270/Q2KW5FVB
More data for this
Ligand-Target Pair