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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Glucose-dependent insulinotropic receptor' and Ligand = 'BDBM50244793'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Glucose-dependent insulinotropic receptor


(Homo sapiens (Human))		BDBM50244793
PNG
(3-fluoro-N-isopropyl-4-(6-(4-(3-isopropyl-1,2,4-ox...)
Show SMILES CC(C)c1nc([o+][n-]1)C1CCN(CC1)c1ncnc(Nc2ccc(cc2F)S(=O)(=O)C(C)C)c1[N+]([O-])=O
Show InChI InChI=1S/C23H28FN7O5S/c1-13(2)20-28-23(36-29-20)15-7-9-30(10-8-15)22-19(31(32)33)21(25-12-26-22)27-18-6-5-16(11-17(18)24)37(34,35)14(3)4/h5-6,11-15H,7-10H2,1-4H3,(H,25,26,27)
PDB

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PC sid
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Similars
Article
PubMed
n/an/an/an/a 7.90n/an/an/an/a



Arena Pharmaceuticals

Curated by ChEMBL


Assay Description
Agonist activity at CPR119 (unknown origin) transfected in Xenopus dermal melanophore assessed as dispersion of melatonin-induced pigmentation

J Med Chem 51: 5172-5 (2008)


Article DOI: 10.1021/jm8006867
BindingDB Entry DOI: 10.7270/Q2KW5FVB
More data for this
Ligand-Target Pair