Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
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Glutamate receptor 2 (Homo sapiens (Human)) | BDBM50355329 (CHEMBL1835336) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem | PDB Article PubMed | 3.15E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Displacement of [3H]AMPA from recombinant GluA2 S1S2J soluble ligand binding domain | J Med Chem 54: 7289-98 (2011) Article DOI: 10.1021/jm200862h BindingDB Entry DOI: 10.7270/Q2QC03WT | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) |