BindingDB logo
myBDB logout
Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Glutamate receptor 2' and Ligand = 'BDBM50494341'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Glutamate receptor 2


(Homo sapiens (Human))		BDBM50494341
PNG
(LY-293,558 | LY-293558 | NGX-424 | TEZAMPANEL)
Show SMILES [H][C@@]12CC[C@H](CCc3nn[nH]n3)C[C@]1([H])C[C@H](NC2)C(O)=O
Show InChI InChI=1S/C13H21N5O2/c19-13(20)11-6-10-5-8(1-3-9(10)7-14-11)2-4-12-15-17-18-16-12/h8-11,14H,1-7H2,(H,19,20)(H,15,16,17,18)/t8-,9+,10-,11+/m1/s1
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
Purchase

PC cid
PC sid
UniChem
Article
PubMed
 3.00E+3n/an/an/an/an/an/an/an/a



Centro de Investigaci�n Lilly

Curated by ChEMBL


Assay Description
Displacement of [3H]AMPA from homomeric recombinant GluA2 receptor (unknown origin)

Bioorg Med Chem Lett 23: 6463-6 (2013)


Article DOI: 10.1016/j.bmcl.2013.09.045
BindingDB Entry DOI: 10.7270/Q2XS5ZBW
More data for this
Ligand-Target Pair