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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Glutamate receptor 4' and Ligand = 'BDBM50112773'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Glutamate receptor 4


(Homo sapiens (Human))		BDBM50112773
PNG
((+/-3b) N-{4'-[1-Methyl-2-(propane-2-sulfonylamino...)
Show SMILES CC(C)S(=O)(=O)NCC(C)c1ccc(cc1)-c1ccc(NC(=O)c2ccccc2)cc1
Show InChI InChI=1S/C25H28N2O3S/c1-18(2)31(29,30)26-17-19(3)20-9-11-21(12-10-20)22-13-15-24(16-14-22)27-25(28)23-7-5-4-6-8-23/h4-16,18-19,26H,17H2,1-3H3,(H,27,28)
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n/an/an/an/a 520n/an/an/an/a



NPS Allelix Corporation

Curated by ChEMBL


Assay Description
Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.

J Med Chem 45: 2101-11 (2002)


BindingDB Entry DOI: 10.7270/Q20R9NRB
More data for this
Ligand-Target Pair