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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Glutamate receptor ionotropic, NMDA 1' and Ligand = 'BDBM50002702'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Glutamate receptor ionotropic, NMDA 1


(RAT)		BDBM50002702
PNG
(7,8-Dichloro-1-trifluoromethyl-5H-[1,2,4]triazolo[...)
Show SMILES FC(F)(F)c1nnc2n1c1cc(Cl)c(Cl)cc1[nH]c2=O
Show InChI InChI=1S/C10H3Cl2F3N4O/c11-3-1-5-6(2-4(3)12)19-7(8(20)16-5)17-18-9(19)10(13,14)15/h1-2H,(H,16,20)
PDB

UniProtKB/SwissProt

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PC cid
PC sid
UniChem

Patents

Similars
PubMed
>1.00E+4n/an/an/an/an/an/an/an/a



Lilly Research Laboratories

Curated by ChEMBL


Assay Description
Displacement of [3H]glycine from glycine site on the NMDA receptor.

J Med Chem 35: 3319-24 (1992)


BindingDB Entry DOI: 10.7270/Q2WM1F13
More data for this
Ligand-Target Pair