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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Glutamate receptor ionotropic, NMDA 1' and Ligand = 'BDBM50056655'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Glutamate receptor ionotropic, NMDA 1


(RAT)		BDBM50056655
PNG
(CHEMBL164295 | N-(7-Chloro-2-oxo-3-phenyl-1,2-dihy...)
Show SMILES CC(=O)Nc1c(-c2ccccc2)c(=O)[nH]c2cc(Cl)ccc12
Show InChI InChI=1S/C17H13ClN2O2/c1-10(21)19-16-13-8-7-12(18)9-14(13)20-17(22)15(16)11-5-3-2-4-6-11/h2-9H,1H3,(H2,19,20,21,22)
PDB

UniProtKB/SwissProt

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PC cid
PC sid
UniChem

Patents

Similars
Article
PubMed
n/an/a 1.47E+4n/an/an/an/an/an/a



Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL


Assay Description
In vitro ability to displace [3H]L-689,560 binding to glycine site on the N-methyl-D-aspartate (NMDA) glutamate receptor 1 from rat cortical membrane...

J Med Chem 40: 754-65 (1997)


Article DOI: 10.1021/jm9605492
BindingDB Entry DOI: 10.7270/Q2J67G1J
More data for this
Ligand-Target Pair