BindingDB logo
myBDB logout
Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Glutamate receptor ionotropic, NMDA 1' and Ligand = 'BDBM50110210'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Glutamate receptor ionotropic, NMDA 1


(RAT)		BDBM50110210
PNG
(8-Chloro-9-nitro-5-oxo-5,6-dihydro-pyrazolo[1,5-c]...)
Show SMILES OC(=O)c1cc2c3cc(c(Cl)cc3[n-]c(=[OH+])n2n1)[N+]([O-])=O
Show InChI InChI=1S/C11H5ClN4O5/c12-5-2-6-4(1-9(5)16(20)21)8-3-7(10(17)18)14-15(8)11(19)13-6/h1-3H,(H2,13,14,17,18,19)
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
CHEMBL
PC cid
PC sid
UniChem

Similars
PubMed
 1.10E+3n/an/an/an/an/an/an/an/a



Universita' di Firenze

Curated by ChEMBL


Assay Description
Percent Inhibition by displacing [3H]-Glycine of N-methyl-D-aspartate glutamate receptor 1 in rat cortical membranes

J Med Chem 45: 1035-44 (2002)


BindingDB Entry DOI: 10.7270/Q2WD3ZW6
More data for this
Ligand-Target Pair