Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Glycogen phosphorylase, muscle form (Oryctolagus cuniculus (rabbit)) | BDBM50263769 ((5S,7R,8S,9S,10R)-8,9,10-Trihydroxy-7-hydroxymethy...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL MMDB PC cid PC sid PDB UniChem Similars | MMDB PDB Article PubMed | 5.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Inhibition of rabbit muscle glycogen phosphorylase b | Bioorg Med Chem Lett 18: 5680-3 (2008) Article DOI: 10.1016/j.bmcl.2008.08.052 BindingDB Entry DOI: 10.7270/Q2571BTV | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Glycogen phosphorylase, muscle form (Homo sapiens (Human)) | BDBM50263769 ((5S,7R,8S,9S,10R)-8,9,10-Trihydroxy-7-hydroxymethy...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL MMDB PC cid PC sid PDB UniChem Similars | MMDB PDB PubMed | 5.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lajos Kossuth University Curated by ChEMBL | Assay Description Inhibitor constant was measured against Muscle phosphorylase b in rabbit | Bioorg Med Chem Lett 9: 1385-90 (1999) BindingDB Entry DOI: 10.7270/Q2W66M82 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Glycogen phosphorylase, muscle form (Oryctolagus cuniculus (rabbit)) | BDBM50263769 ((5S,7R,8S,9S,10R)-8,9,10-Trihydroxy-7-hydroxymethy...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL MMDB PC cid PC sid PDB UniChem Similars | MMDB PDB Article PubMed | 5.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | 6.8 | n/a |
University of Debrecen Curated by ChEMBL | Assay Description Inhibition of rabbit muscle glycogen phosphorylase b assessed as inorganic phosphate release at pH 6.8 | Bioorg Med Chem 20: 1801-16 (2012) Article DOI: 10.1016/j.bmc.2011.12.059 BindingDB Entry DOI: 10.7270/Q2SN09DD | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Glycogen phosphorylase, muscle form (Oryctolagus cuniculus (rabbit)) | BDBM50263769 ((5S,7R,8S,9S,10R)-8,9,10-Trihydroxy-7-hydroxymethy...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL MMDB PC cid PC sid PDB UniChem Similars | MMDB PDB Article PubMed | 5.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ Claude Bernard Lyon 1 Curated by ChEMBL | Assay Description Competitive inhibition of rabbit skeletal muscle glycogen phosphorylase b | Eur J Med Chem 108: 444-54 (2016) Article DOI: 10.1016/j.ejmech.2015.12.004 BindingDB Entry DOI: 10.7270/Q2QR500M | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Glycogen phosphorylase, muscle form (Homo sapiens (Human)) | BDBM50263769 ((5S,7R,8S,9S,10R)-8,9,10-Trihydroxy-7-hydroxymethy...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL MMDB PC cid PC sid PDB UniChem Similars | MMDB PDB PubMed | 1.09E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lajos Kossuth University Curated by ChEMBL | Assay Description Inhibitor constant was measured against Muscle phosphorylase a in rabbit | Bioorg Med Chem Lett 9: 1385-90 (1999) BindingDB Entry DOI: 10.7270/Q2W66M82 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) |