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Found 1 hit Enz. Inhib. hit(s) with Target = 'Gonadotropin-releasing hormone receptor' and Ligand = 'BDBM50097016'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Gonadotropin-releasing hormone receptor


(Rattus norvegicus)		BDBM50097016
PNG
(4-({2-[2-(3,4-Dimethoxy-phenyl)-1H-indol-3-yl]-eth...)
Show SMILES COc1ccc(cc1OC)-c1[nH]c2ccccc2c1CCNCc1ccc(O)cc1
Show InChI InChI=1S/C25H26N2O3/c1-29-23-12-9-18(15-24(23)30-2)25-21(20-5-3-4-6-22(20)27-25)13-14-26-16-17-7-10-19(28)11-8-17/h3-12,15,26-28H,13-14,16H2,1-2H3
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
CHEMBL
PC cid
PC sid
UniChem

Similars
PubMed
n/an/a 2.00E+4n/an/an/an/an/an/a



Merck Research Laboratories

Curated by ChEMBL


Assay Description
Ability to displace [125I]- - radio-labeled buserelin from rat Gonadotropin-releasing hormone receptor

Bioorg Med Chem Lett 11: 509-13 (2001)


BindingDB Entry DOI: 10.7270/Q2BR8RF8
More data for this
Ligand-Target Pair