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Found 1 hit Enz. Inhib. hit(s) with Target = 'Hepatocyte growth factor receptor' and Ligand = 'BDBM50152679'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Hepatocyte growth factor receptor


(Homo sapiens (Human))		BDBM50152679
PNG
(CHEMBL3780556)
Show SMILES COc1cc2c(Oc3ccc(NC(=O)c4c(Cl)c5ccccc5n(-c5ccc(F)cc5)c4=O)cc3F)ccnc2cc1OCCCN1CCCC1
Show InChI InChI=1S/C39H33ClF2N4O5/c1-49-34-22-28-30(23-35(34)50-20-6-19-45-17-4-5-18-45)43-16-15-32(28)51-33-14-11-25(21-29(33)42)44-38(47)36-37(40)27-7-2-3-8-31(27)46(39(36)48)26-12-9-24(41)10-13-26/h2-3,7-16,21-23H,4-6,17-20H2,1H3,(H,44,47)
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PC cid
PC sid
UniChem
Article
PubMed
n/an/a 13n/an/an/an/an/an/a



Jiangxi Science and Technology Normal University

Curated by ChEMBL


Assay Description
Inhibition of cMet (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assay

Bioorg Med Chem Lett 26: 1794-8 (2016)


Article DOI: 10.1016/j.bmcl.2016.02.037
BindingDB Entry DOI: 10.7270/Q2TT4ST4
More data for this
Ligand-Target Pair