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Found 1 hit Enz. Inhib. hit(s) with Target = 'Histamine H3 receptor' and Ligand = 'BDBM50071345'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Histamine H3 receptor


(GUINEA PIG)		BDBM50071345
PNG
(4-Chloro-N-[3-(1H-imidazol-4-yl)-propyl]-benzenesu...)
Show SMILES Clc1ccc(cc1)S(=O)(=O)NCCCc1cnc[nH]1
Show InChI InChI=1S/C12H14ClN3O2S/c13-10-3-5-12(6-4-10)19(17,18)16-7-1-2-11-8-14-9-15-11/h3-6,8-9,16H,1-2,7H2,(H,14,15)
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
CHEMBL
PC cid
PC sid
UniChem

Similars
PubMed
 380n/an/an/an/an/an/an/an/a



Schering-Plough Research Institute

Curated by ChEMBL


Assay Description
Inhibition of [3H]-Nalpha-methylhistamine binding to H3 receptor in guinea-pig brain membranes

Bioorg Med Chem Lett 8: 2157-62 (1999)


BindingDB Entry DOI: 10.7270/Q23T9GCZ
More data for this
Ligand-Target Pair