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Found 1 hit Enz. Inhib. hit(s) with Target = 'Histamine H3 receptor' and Ligand = 'BDBM50148119'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Histamine H3 receptor


(Rattus norvegicus (rat))		BDBM50148119
PNG
(3-[3-(1H-Imidazol-4-yl)-propoxy]-benzonitrile | CH...)
Show SMILES N#Cc1cccc(OCCCc2cnc[nH]2)c1
Show InChI InChI=1S/C13H13N3O/c14-8-11-3-1-5-13(7-11)17-6-2-4-12-9-15-10-16-12/h1,3,5,7,9-10H,2,4,6H2,(H,15,16)
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Similars
Article
PubMed
 108n/an/an/an/an/an/an/an/a



University College London

Curated by ChEMBL


Assay Description
In vitro inhibitory activity against against histamine H3 receptor using [3H]-Histamine as radioligand from rat cerebral cortex synaptosomes

J Med Chem 47: 3264-74 (2004)


Article DOI: 10.1021/jm031141p
BindingDB Entry DOI: 10.7270/Q2F47NK5
More data for this
Ligand-Target Pair