Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50377992 (CHEMBL1202070) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 49 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Jagiellonian University Medical College Curated by ChEMBL | Assay Description Displacement of [125I]Iodoproxyfran from human histamine H3 receptor expressed in HEK293 cells | Bioorg Med Chem 17: 3037-42 (2009) Article DOI: 10.1016/j.bmc.2009.03.014 BindingDB Entry DOI: 10.7270/Q2SF2X3H | |||||||||||
More data for this Ligand-Target Pair |