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Found 1 hit Enz. Inhib. hit(s) with Target = 'Histamine H3 receptor' and Ligand = 'BDBM50462834'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Histamine H3 receptor


(Rattus norvegicus (rat))		BDBM50462834
PNG
(CHEMBL4250218)
Show SMILES Clc1ccc(Cc2noc(CCN3CCCCC3)n2)cc1
Show InChI InChI=1S/C16H20ClN3O/c17-14-6-4-13(5-7-14)12-15-18-16(21-19-15)8-11-20-9-2-1-3-10-20/h4-7H,1-3,8-12H2
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PC cid
PC sid
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Article
PubMed
 126n/an/an/an/an/an/an/an/a



Heinrich Heine University D£sseldorf

Curated by ChEMBL


Assay Description
Displacement of [3H](R)-alpha-methylhistamine from histamine H3 receptor in rat brain membranes

Bioorg Med Chem 26: 4034-4046 (2018)


Article DOI: 10.1016/j.bmc.2018.06.028
BindingDB Entry DOI: 10.7270/Q29026FG
More data for this
Ligand-Target Pair