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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Histone acetyltransferase KAT6A [507-778]' and Ligand = 'BDBM534161'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Histone acetyltransferase KAT6A [507-778]


(Homo sapiens)		BDBM534161
PNG
(6-Cyclopropyl-N-[2-(cyclopropylmethoxy)-5-isopropy...)
Show SMILES CC(C)c1ccc(OCC2CC2)c(c1)S(=O)(=O)NC(=O)c1cc2c(F)cc(cc2o1)C1CC1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
WIPO WO2022081842
n/an/a 3.01n/an/an/an/an/an/a


TBA

Assay Description
 Kat6a inhibitory activities of the compounds described in the present invention were quantified using a Fluorescence Resonance Energy Transfer (TR-F...

Citation and Details

BindingDB Entry DOI: 10.7270/Q2VM4GFQ
More data for this
Ligand-Target Pair