Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Histone acetyltransferase KAT8 (Homo sapiens (Human)) | BDBM50581154 (CHEMBL5090533) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human MOF using AcCoA and H4 peptide as substrate incubated for 12 min at room temperature relative to control | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00141 BindingDB Entry DOI: 10.7270/Q2XK8KFR | |||||||||||
More data for this Ligand-Target Pair |