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Found 1 hit Enz. Inhib. hit(s) with Target = 'Histone-lysine N-methyltransferase EHMT2' and Ligand = 'BDBM50324901'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Histone-lysine N-methyltransferase EHMT2


(Homo sapiens (Human))		BDBM50324901
PNG
(2,2-dihydroxy-1H-indene-1,3(2H)-dione | CHEMBL1221...)
Show SMILES OC1(O)C(=O)c2ccccc2C1=O
Show InChI InChI=1S/C9H6O4/c10-7-5-3-1-2-4-6(5)8(11)9(7,12)13/h1-4,12-13H
PDB

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CHEMBL
MCE
PC cid
PC sid
UniChem

Patents
Article
PubMed
n/an/a 5.40E+4n/an/an/an/an/an/a



Radboud University

Curated by ChEMBL


Assay Description
Inhibition of wild type recombinant human histone lysine methyltransferase G9a (913 to 1193 residues) expressed in Escherichia coli Rosetta BL21 DE3 ...

Bioorg Med Chem Lett 28: 1234-1238 (2018)


Article DOI: 10.1016/j.bmcl.2018.02.043
BindingDB Entry DOI: 10.7270/Q24Q7XKJ
More data for this
Ligand-Target Pair