Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Homeodomain-interacting protein kinase 3 (Homo sapiens (Human)) | BDBM50335638 (5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | n/a | n/a | 45 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of recombinant human HIPK3 in presence of ATP at Km concentration by radiometric filter-binding assay | Citation and Details Article DOI: 10.1016/j.ejmech.2020.112770 BindingDB Entry DOI: 10.7270/Q2DN48PP | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Homeodomain-interacting protein kinase 3 (Homo sapiens (Human)) | BDBM50335638 (5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | n/a | n/a | 45 | n/a | n/a | n/a | n/a | n/a | n/a |
Cylene Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of human recombinant HIPK3 by radiometric assay | J Med Chem 54: 635-54 (2011) Article DOI: 10.1021/jm101251q BindingDB Entry DOI: 10.7270/Q2J67H7N | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) |