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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Importin subunit alpha-1' and Ligand = 'BDBM75081'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Importin subunit alpha-1


(Homo sapiens (Human))		BDBM75081
PNG
(2-[2-(3-ethanoylphenoxy)ethanoyl-methyl-amino]-N-(...)
Show SMILES CN(CC(=O)Nc1ccc(F)cc1)C(=O)COc1cccc(c1)C(C)=O
Show InChI InChI=1S/C19H19FN2O4/c1-13(23)14-4-3-5-17(10-14)26-12-19(25)22(2)11-18(24)21-16-8-6-15(20)7-9-16/h3-10H,11-12H2,1-2H3,(H,21,24)
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n/an/an/an/a>5.00E+5n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...

PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair