Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Integrin alpha-5/beta-1 (Homo sapiens (Human)) | BDBM50074659 ((S)-2-[(S)-3-Carboxy-2-((S)-4-methyl-2-{2-[4-(3-o-...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Biogen Inc. Curated by ChEMBL | Assay Description Inhibition of integrin alpha5-beta1 adhesion to K562 cells | J Med Chem 42: 920-34 (1999) Article DOI: 10.1021/jm980673g BindingDB Entry DOI: 10.7270/Q2P26XBF | |||||||||||
More data for this Ligand-Target Pair |