Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Kappa-type opioid receptor (Cavia porcellus (domestic guinea pig)) | BDBM50491880 (CHEMBL2387724) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 0.150 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Displacement of [3H]U-69,593 from kappa opioid receptor in guinea pig cerebellum | Bioorg Med Chem 21: 3032-50 (2013) Article DOI: 10.1016/j.bmc.2013.03.026 BindingDB Entry DOI: 10.7270/Q2JQ13XJ | |||||||||||
More data for this Ligand-Target Pair |