Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
KiSS-1 receptor (Homo sapiens (Human)) | BDBM50082076 (CHEMBL3422409) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.600 | n/a | n/a | n/a | n/a |
UMR7247; Universit£ Fran£ois Rabelais Tours; IFCE) Curated by ChEMBL | Assay Description Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 ... | J Med Chem 58: 3459-70 (2015) Article DOI: 10.1021/jm5019675 BindingDB Entry DOI: 10.7270/Q2JD4ZHJ | |||||||||||
More data for this Ligand-Target Pair |