Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Leukotriene B4 receptor 1 (Homo sapiens (Human)) | BDBM50174606 (CHEMBL384950 | HYNIC Analogue) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 44 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Bristol-Myers Squibb Medical Imaging Curated by ChEMBL | Assay Description Inhibitory concentration against human leukotriene B4 receptor using competing agent [111In]-(17)] as radioligand in pH 7.2 buffer, for 1 h at 37 deg... | J Med Chem 48: 6442-53 (2005) Article DOI: 10.1021/jm050383h BindingDB Entry DOI: 10.7270/Q2959H33 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Leukotriene B4 receptor 1 (Homo sapiens (Human)) | BDBM50174606 (CHEMBL384950 | HYNIC Analogue) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 45 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Bristol-Myers Squibb Medical Imaging Curated by ChEMBL | Assay Description Inhibitory concentration against human leukotriene B4 receptor using competing agent [3H]-LTB4 as radioligand in pH 7.2 buffer upon incubation for 1 ... | J Med Chem 48: 6442-53 (2005) Article DOI: 10.1021/jm050383h BindingDB Entry DOI: 10.7270/Q2959H33 | |||||||||||
More data for this Ligand-Target Pair |