Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Low molecular weight phosphotyrosine protein phosphatase (Homo sapiens (Human)) | BDBM50118216 ((4-formyl-5-hydroxy-6-methylpyridin-3-yl)methyl di...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 1.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Saint John's University Curated by ChEMBL | Assay Description Competitive inhibition of LMW-PTP isoform A (unknown origin) | Bioorg Med Chem Lett 30: (2020) Article DOI: 10.1016/j.bmcl.2020.127342 BindingDB Entry DOI: 10.7270/Q2FJ2MBV | |||||||||||
More data for this Ligand-Target Pair |