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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Lysine-specific demethylase 4C' and Ligand = 'BDBM347135'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Lysine-specific demethylase 4C


(Homo sapiens (Human))		BDBM347135
PNG
(2-(4-((cyclopropylmethyl)(3-(4-methyl piperazin-1-...)
Show SMILES CN1CCN(CC1)c1cccc(c1)N(CC1CC1)c1ccc(Oc2nc(O)c3ccncc3n2)cc1
Show InChI InChI=1S/C28H30N6O2/c1-32-13-15-33(16-14-32)22-3-2-4-23(17-22)34(19-20-5-6-20)21-7-9-24(10-8-21)36-28-30-26-18-29-12-11-25(26)27(35)31-28/h2-4,7-12,17-18,20H,5-6,13-16,19H2,1H3,(H,30,31,35)
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US Patent
n/an/a<100n/an/an/an/an/an/a



CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate-format under the following reaction conditions: 0.3 ...

US Patent US10202381 (2019)


BindingDB Entry DOI: 10.7270/Q2SX6GBM
More data for this
Ligand-Target Pair