BindingDB PrimarySearch

Found 1 hit Enz. Inhib. hit(s) with Target = 'Lysine-specific demethylase 5A' and Ligand = 'BDBM320395'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Lysine-specific demethylase 5A (Homo sapiens (Human))	BDBM320395 (2-[hydroxy(oxan-4-yl)methyl]- 1H-pyrrolo[3,2-b]pyr...) Show SMILES OC(C1CCOCC1)c1cc2nccc(C(O)=O)c2[nH]1 Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<100	n/a	n/a	n/a	n/a	n/a	n/a
Celgene Quantical Research, Inc. US Patent					Assay Description The enzymatic assay of Jarid1A activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test c...				US Patent US9738637 (2017) BindingDB Entry DOI: 10.7270/Q2VD71K6
Celgene Quantical Research, Inc. US Patent					More data for this Ligand-Target Pair