BindingDB PrimarySearch

Found 2 hits Enz. Inhib. hit(s) with Target = 'Mas-related G-protein coupled receptor member X1' and Ligand = 'BDBM50340753'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Mas-related G-protein coupled receptor member X1 (Homo sapiens (Human))	BDBM50340753 (2-(4-(2-(4-chlorophenethylamino)pyrimidin-4-yl)pip...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	14	n/a	n/a	n/a	n/a	n/a	n/a
AstraZeneca R&D Montreal Curated by ChEMBL					Assay Description Antagonist activity at SNSR4 in human HEK293 cells by FLIPR assay				Bioorg Med Chem Lett 21: 2102-5 (2011) Article DOI: 10.1016/j.bmcl.2011.01.138 BindingDB Entry DOI: 10.7270/Q2D21XW7
AstraZeneca R&D Montreal Curated by ChEMBL					More data for this Ligand-Target Pair
Mas-related G-protein coupled receptor member X1 (Homo sapiens (Human))	BDBM50340753 (2-(4-(2-(4-chlorophenethylamino)pyrimidin-4-yl)pip...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	50	n/a	n/a	n/a	n/a	n/a	n/a
Johns Hopkins University Curated by ChEMBL					Assay Description Antagonist activity at human MrgX1 transfected in HEK293 cells by FLIPR assay				Bioorg Med Chem 22: 5831-7 (2014) Article DOI: 10.1016/j.bmc.2014.09.025 BindingDB Entry DOI: 10.7270/Q27P92CV
Johns Hopkins University Curated by ChEMBL					More data for this Ligand-Target Pair