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Found 1 hit Enz. Inhib. hit(s) with Target = 'Melanin-concentrating hormone receptor 1' and Ligand = 'BDBM50107738'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM50107738
PNG
(CHEMBL3600818)
Show SMILES CCNC(=O)N(C)Cc1ccc(CCNC(=O)c2ccc(cc2F)-c2ccc(Cl)cc2)cc1
Show InChI InChI=1S/C26H27ClFN3O2/c1-3-29-26(33)31(2)17-19-6-4-18(5-7-19)14-15-30-25(32)23-13-10-21(16-24(23)28)20-8-11-22(27)12-9-20/h4-13,16H,3,14-15,17H2,1-2H3,(H,29,33)(H,30,32)
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Article
PubMed
n/an/a 36n/an/an/an/an/an/a



Boehringer Ingelheim Pharma GmbH& Co. KG

Curated by ChEMBL


Assay Description
Displacement of [125I]-MCH from human MCHR1 expressed in CHO/Galpha16 cell membranes by scintillation counting method

Bioorg Med Chem Lett 25: 3264-9 (2015)


Article DOI: 10.1016/j.bmcl.2015.05.077
BindingDB Entry DOI: 10.7270/Q25D8TMB
More data for this
Ligand-Target Pair