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Found 1 hit Enz. Inhib. hit(s) with Target = 'Melanin-concentrating hormone receptor 1' and Ligand = 'BDBM50152463'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM50152463
PNG
(8-[3-(2,2-Difluoro-benzo[1,3]dioxol-5-ylamino)-pro...)
Show SMILES Nc1ccc2cccc(OCCCNc3ccc4OC(F)(F)Oc4c3)c2n1
Show InChI InChI=1S/C19H17F2N3O3/c20-19(21)26-14-7-6-13(11-16(14)27-19)23-9-2-10-25-15-4-1-3-12-5-8-17(22)24-18(12)15/h1,3-8,11,23H,2,9-10H2,(H2,22,24)
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Similars
Article
PubMed
n/an/a 1n/an/an/an/an/an/a



Abbott Laboratories

Curated by ChEMBL


Assay Description
Concentration required to inhibit binding of [125I]-MCH radioligand to human Melanin-concentrating hormone receptor 1 in IMR-32 I3.4.2 cell membranes

Bioorg Med Chem Lett 14: 4879-82 (2004)


Article DOI: 10.1016/j.bmcl.2004.07.034
BindingDB Entry DOI: 10.7270/Q2M32V61
More data for this
Ligand-Target Pair