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Found 1 hit Enz. Inhib. hit(s) with Target = 'Melanin-concentrating hormone receptor 1' and Ligand = 'BDBM50152469'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM50152469
PNG
(CHEMBL182575 | N-[3-(2-{[5-(4-Chloro-phenyl)-furan...)
Show SMILES Clc1ccc(cc1)-c1ccc(CNc2ccc3cccc(OCCCNC(=O)c4cccc(c4)C#N)c3n2)o1
Show InChI InChI=1S/C31H25ClN4O3/c32-25-11-8-22(9-12-25)27-14-13-26(39-27)20-35-29-15-10-23-5-2-7-28(30(23)36-29)38-17-3-16-34-31(37)24-6-1-4-21(18-24)19-33/h1-2,4-15,18H,3,16-17,20H2,(H,34,37)(H,35,36)
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n/an/a 2n/an/an/an/an/an/a



Abbott Laboratories

Curated by ChEMBL


Assay Description
Concentration required to inhibit binding of [125I]-MCH radioligand to human Melanin-concentrating hormone receptor 1 in IMR-32 I3.4.2 cell membranes

Bioorg Med Chem Lett 14: 4879-82 (2004)


Article DOI: 10.1016/j.bmcl.2004.07.034
BindingDB Entry DOI: 10.7270/Q2M32V61
More data for this
Ligand-Target Pair