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Found 1 hit Enz. Inhib. hit(s) with Target = 'Melanin-concentrating hormone receptor 1' and Ligand = 'BDBM50191760'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM50191760
PNG
(CHEMBL216038 | N-(3-dimethylaminomethyl-quinolin-8...)
Show SMILES CN(C)Cc1cnc2c(CNC(=O)c3ccc(nc3)-c3ccc(F)cc3)cccc2c1
Show InChI InChI=1S/C25H23FN4O/c1-30(2)16-17-12-19-4-3-5-20(24(19)28-13-17)14-29-25(31)21-8-11-23(27-15-21)18-6-9-22(26)10-7-18/h3-13,15H,14,16H2,1-2H3,(H,29,31)
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Similars
Article
PubMed
 414n/an/an/an/an/an/an/an/a



Procter and Gamble Pharmaceuticals Inc.

Curated by ChEMBL


Assay Description
Binding affinity to MCHR1 by radioligand binding assay

Bioorg Med Chem Lett 16: 5207-11 (2006)


Article DOI: 10.1016/j.bmcl.2006.07.006
BindingDB Entry DOI: 10.7270/Q2SX6CV3
More data for this
Ligand-Target Pair