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Found 1 hit Enz. Inhib. hit(s) with Target = 'Melanin-concentrating hormone receptor 1' and Ligand = 'BDBM50301083'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM50301083
PNG
(4-(4-fluorobenzyloxy)-1-(3-(2-(pyrrolidin-1-yl)eth...)
Show SMILES Fc1ccc(COc2ccn(Cc3cccc(OCCN4CCCC4)c3)c(=O)c2)cc1
Show InChI InChI=1S/C25H27FN2O3/c26-22-8-6-20(7-9-22)19-31-24-10-13-28(25(29)17-24)18-21-4-3-5-23(16-21)30-15-14-27-11-1-2-12-27/h3-10,13,16-17H,1-2,11-12,14-15,18-19H2
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Article
PubMed
n/an/a 29n/an/an/an/an/an/a



Tsukuba Research Institute

Curated by ChEMBL


Assay Description
Antagonistic activity against MCH1R expressed on CHOK1 cells assessed as intracellular calcium mobilization by FLIPR

Bioorg Med Chem Lett 19: 5186-90 (2009)


Article DOI: 10.1016/j.bmcl.2009.07.023
BindingDB Entry DOI: 10.7270/Q2G44QCG
More data for this
Ligand-Target Pair