Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Melanocortin receptor 3 (Homo sapiens (Human)) | BDBM50323150 (CHEMBL1209253 | N-(2-(4-((3S,4R)-1-tert-butyl-4-(2...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [125I]NDP-alpha-MSH from human MC3 receptor expressed in CHO cells | Bioorg Med Chem Lett 20: 4483-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.038 BindingDB Entry DOI: 10.7270/Q2C829GJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Homo sapiens (Human)) | BDBM50323150 (CHEMBL1209253 | N-(2-(4-((3S,4R)-1-tert-butyl-4-(2...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.80E+3 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Agonist activity at human MC3 receptor expressed in CHO cells assessed as increase of alpha-MSH-induced cAMP accumulation | Bioorg Med Chem Lett 20: 4483-6 (2010) Article DOI: 10.1016/j.bmcl.2010.06.038 BindingDB Entry DOI: 10.7270/Q2C829GJ | |||||||||||
More data for this Ligand-Target Pair |