Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50453139 (CHEMBL4205548) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 630 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Naples "Federico II" Curated by ChEMBL | Assay Description Displacement of [125I]-NDP-alpha-MSH from human MC5R expressed in HEK293 cells after 40 mins by gamma counting method | J Med Chem 61: 4263-4269 (2018) Article DOI: 10.1021/acs.jmedchem.8b00488 BindingDB Entry DOI: 10.7270/Q22J6FF7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50453139 (CHEMBL4205548) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.90 | n/a | n/a | n/a | n/a |
University of Naples "Federico II" Curated by ChEMBL | Assay Description Agonist activity at human MC5R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 mins | J Med Chem 61: 4263-4269 (2018) Article DOI: 10.1021/acs.jmedchem.8b00488 BindingDB Entry DOI: 10.7270/Q22J6FF7 | |||||||||||
More data for this Ligand-Target Pair |