Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Metabotropic glutamate receptor 1 (RAT) | BDBM50288204 ((2S,3S)-3-Carboxymethyl-azetidine-2-carboxylic aci...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 1.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Compound was tested in vitro for binding affinity against mGluR1a metabotropic glutamate receptor, using [3H]-glutamate as the radioligand. | Bioorg Med Chem Lett 6: 2559-2564 (1996) Article DOI: 10.1016/0960-894X(96)00464-7 BindingDB Entry DOI: 10.7270/Q2HX1CN1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 1 (Homo sapiens (Human)) | BDBM50288204 ((2S,3S)-3-Carboxymethyl-azetidine-2-carboxylic aci...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | n/a | n/a | 2.10E+5 | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Compound was tested for its agonist activity against mGluR1a receptor in CHO cells. | Bioorg Med Chem Lett 6: 2559-2564 (1996) Article DOI: 10.1016/0960-894X(96)00464-7 BindingDB Entry DOI: 10.7270/Q2HX1CN1 | |||||||||||
More data for this Ligand-Target Pair |