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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 4' and Ligand = 'BDBM50323571'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Metabotropic glutamate receptor 4


(Homo sapiens (Human))		BDBM50323571
PNG
(4-(3-fluorostyryl)pyrimidin-2-amine | CHEMBL120966...)
Show SMILES Nc1nccc(\C=C\c2cccc(F)c2)n1
Show InChI InChI=1S/C12H10FN3/c13-10-3-1-2-9(8-10)4-5-11-6-7-15-12(14)16-11/h1-8H,(H2,14,15,16)/b5-4+
PDB

UniProtKB/SwissProt

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CHEMBL
PC cid
PC sid
UniChem

Similars
Article
PubMed
n/an/an/an/a 4.50E+3n/an/an/an/a



Evotec (UK) Ltd

Curated by ChEMBL


Assay Description
Positive allosteric modulation of human mGluR4 expressed in CHO-K1 cells assessed as decrease in forskolin-induced intracellular cAMP accumulation af...

Bioorg Med Chem Lett 20: 4901-5 (2010)


Article DOI: 10.1016/j.bmcl.2010.06.078
BindingDB Entry DOI: 10.7270/Q2X34XN7
More data for this
Ligand-Target Pair